Publications 2021

  • Sulfoximines with α‐Ketoester Functionalities at Nitrogen from Cyanoacetates and Air
    C. Wang, H. Wang, C. Bolm, Adv. Synth. Catal. 2021, 363, 747–750.
  • NH-sulfoximine: A novel pharmacological inhibitor of the mitochondrial F1Fo‐ATPase, which suppresses viability of cancerous cells
    D. Strobbe, R. Pecorari, O. Conte, A. Minutolo, C. M. M. Hendriks, S. Wiezorek, D. Faccenda, R. Abeti, C. Montesano, C. Bolm, M. Campanella, Br. J. Pharmacol. 2021, 178, 298–311.
  • 1,2-Benzothiazine Derivatives from Sulfonimidamides by Metal-Catalyzed Annulation Reactions in Solution and under Solvent-Free Mechanochemical Conditions
    J.‐H. Schöbel, P. Elbers, K.‐N. Truong, K. Rissanen, C. Bolm, Adv. Synth. Catal. 2021, 363, 1322–1329.
  • Palladium‐Catalyzed Carbonylation in the Synthesis of N‐Ynonylsulfoximines
    D. Ma, C. Wang, D. Kong, Y. Tu, P. Shi, C. Bolm, Adv. Synth. Catal. 2021, 363, 1330–1334.
  • 2,3-Dihydro-1,2,6-thiadiazine 1-Oxides by Biginelli-Type Reactions with Sulfonimidamides under Mechanochemical Conditions
    F. Krauskopf, K.‐N. Truong, K. Rissanen, C. Bolm, Org. Lett. 2021, 23, 2699–2703.
  • 2-Sulfoximidoyl Acetic Acids from Multicomponent Petasis Reactions and Their Use as Building Blocks in Syntheses of Sulfoximine Benzodiazepine Analogues
    R. Hommelsheim, H. M. Núñez Ponce, K.‐N. Truong, K. Rissanen, C. Bolm, Org. Lett. 2021, 23, 3415–3420.
  • Bromodomain Inhibitors
    C. Bolm, M. Frings, J.-H. Schöbel, N. Chatain, B. Altenburg, G. Rossetti, J. Gossen, S. Koschmieder, Patent application, WO2021083879 (A1), May 06, 2021.
    For additional information, please see here.
  • Regio- and Stereoselective Chloro Sulfoximidations of Terminal Aryl Alkynes Enabled by Copper Catalysis and Visible Light
    P. Shi, Y. Tu, D. Zhang, C. Wang, K.‐N. Truong, K. Rissanen, C. Bolm, Adv. Synth. Catal. 2021, 363, 2552–2556.
  • Visible light-promoted NH-halogenation of sulfoximines with dichloromethane or dibromomethane
    C. Wang, P. Shi, C. Bolm, Org. Chem. Front. 2021, 8, 2919–2923.
  • Selected applications of Meldrum's acid – a tutorial
    F. Brosge, P. Singh, F. Almqvist, C. Bolm, Org. Biomol. Chem. 2021, 19, 5014–5027.
  • Investigation of isomerization of dexibuprofen in a ball mill using chiral capillary electrophoresis
    J. Urlaub, R. P. Kaiser, O. Scherf‐Clavel, C. Bolm, U. Holzgrabe, Electrophoresis 2021, 10.1002/elps.202000307.
  • Photochemistry of N-Phenyl Dibenzothiophene Sulfoximine
    A. Isor, R. Hommelsheim, G. W. Cone, M. Frings, J. T. Petroff II, C. Bolm, R. D. McCulla, Photochem. Photobiol. 2021, 10.1111/php.13456.