Publications 2024

  • Mechanochemical Iron-Catalyzed Nitrene Transfer Reactions: Direct Synthesis of N-Acyl Sulfonimidamides from Sulfinamides and Dioxazolones
    S. Pan, F. F. Mulks, P. Wu, K. Rissanen, C. Bolm, Angew. Chem. Int. Ed. 2024, 63, e202316702.
  • Halogen bonding and mechanochemistry combined: synthesis, characterization, and application of N-iodosaccharin pyridine complexes
    C. Schumacher, K.-N. Truong, J. S. Ward, R. Puttreddy, A. Rajala, E. Lassila, C. Bolm, K. Rissanen, Org. Chem. Front. 2024, 11, 781–795.
    Also published as a preprint at ChemRxiv.
  • Microbially-conjugated bile salts found in human bile activate the bile salt receptors TGR5 and FXR
    Ü. Ay, M. Leníček, R. S. Haider, A. Classen, H. van Eijk, K. V. K. Koelfat, G. van der Kroft, U. P. Neumann, C. Hoffmann, C. Bolm, S. W. M. Olde Damink, F. G. Schaap, Hepatol. Commun. 2024, 8, e0383.
    Also published as a preprint at BioRxiv.
  • Unexpected Single-Ligand Occupancy and Negative Cooperativity in the SARS-CoV-2 Main Protease
    S. Albani, E. Costanzi, G. L. Hoang, M. Kuzikov, M. Frings, N. Ansari, N. Demitri, T. T. Nguyen, V. Rizzi, J. B. Schulz, C. Bolm, A. Zaliani, P. Carloni, P. Storici, G. Rossetti, J. Chem. Inf. Model. 2024, 64, 892–904.
    Also published as a preprint at ChemRxiv.
  • Rhodium(II)-Catalyzed N–H Insertions of Carbenes under Mechanochemical Conditions
    S. Biswas, C. Bolm, Org. Lett. 2024, 26, 1511–1516.
  • Palladium-Catalyzed Domino Reaction for the Synthesis of 3-Amino 1,2,4-Benzothiadiazine 1,1-Dioxides
    R. Hommelsheim, R. van Nahl, L. M. Hanek, J. S. Ward, K. Rissanen, C. Bolm, Adv. Synth. Catal. 2024, 366, 717–724.
  • Diversification of NH-Aryl Sulfoximines through Iridium-Catalyzed ortho- and meta-Selective C–H Borylation
    P. van Bonn, S. Soerensen, N. Schmitz, C. Bolm, Adv. Synth. Catal. 2024, 366, 725–732.
  • Synthesis of α-ketothioamides with elemental sulfur under solvent-free conditions in a mixer mill
    C. C. Sahu, S. Biswas, R. Hommelsheim, C. Bolm, RSC Mechanochem. 2024, 1, 38–42.
  • Azasulfur(IV) derivatives of sulfite and sulfinate esters by formal S–S bond insertion of dichloramines
    P. Wu, J. Demaerel, B. J. Statham, C. Bolm, Chem. Sci. 202415, 5333–5339.
  • Mechanochemical Mitsunobu Reactions
    M. T. J. Williams, L. Adarve Cardona, C. Bolm, Adv. Synth. Catal. 2024, 10.1002/adsc.202400296.
  • Synthesis of Benzo[e][1,4,3]oxathiazin-3-one 1-Oxides from NH-S-(2-Hydroxyaryl)sulfoximines
    K. Periasamy, P. van Bonn, R. Tschekorsky Orloff, N. Völcker, Q. Lu, K. Rissanen, C. Bolm, J. Org. Chem. 2024, 10.1021/acs.joc.4c00712.